发明名称 Salts of avermectins substituted in the 4″-position and having pesticidal properties
摘要 A compound of formula wherein X− is an anion; n is 1, 2, 3 or 4; R1 is C1-C12alkyl, C3-C8cycloalkyl; or C2-C12alkenyl; R2 is hydrogen, unsubstituted or substituted C1-C12alkyl or C2-C12alkenyl; R3 is hydrogen, unsubstituted or substituted C1-C12alkyl, C3-C12cycloalkyl, C2-C12alkenyl; or C2-C12alkynyl; or R2 and R3 together are an alkylene or alkenylene bridge; and, where applicable, E/Z isomers, E/Z isomeric mixtures and/or tautomers; with the proviso that R1 is not sec-butyl or isopropyl when R2 is H and R3 is methyl; and, where applicable, their possible tautomers; a process for the preparation of those compounds and their tautomers and the use thereof; pesticidal compositions in which the active ingredient has been selected from those compounds and their tautomers; and a process for the preparation of those compositions and the use thereof; intermediates, in free form or in salt form, for the preparation of those compounds and, where applicable, their tautomers, in free form or in salt form, are described.
申请公布号 US7678773(B2) 申请公布日期 2010.03.16
申请号 US20050319687 申请日期 2005.12.28
申请人 MERIAL LIMITED 发明人 PITTERNA THOMAS
分类号 A61K31/70;C07H17/08;A01N43/90;C07H19/01 主分类号 A61K31/70
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