发明名称 |
TRIAZOLE COMPOUNDS AND USES RELATED THERETO |
摘要 |
The present invention provides a triazole compound of the following formula: a prodrug thereof or a pharmaceutically acceptable salt thereof. The above-mentioned triazole compound has superior HSD1 inhibitory activity, and is useful as an HSD1 inhibitor, a therapeutic drug of diabetes or a therapeutic drug of obesity or a therapeutic drug of metabolic syndrome.
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申请公布号 |
US2010062972(A1) |
申请公布日期 |
2010.03.11 |
申请号 |
US20090621922 |
申请日期 |
2009.11.19 |
申请人 |
AMGEN INC. |
发明人 |
POWERS JAY P.;CARDOZO MARIO G.;GOTO HIROYUKI;HARADA KAZUHITO;IMAMURA KATSUAKI;KAKUTANI MAKOTO;MATSUDA ISAMU;OHE YASUHIRO;YATA SHINJI |
分类号 |
A61K31/4196;A61K;A61K31/18;A61K31/422;A61K31/438;A61K31/445;A61K31/454;A61K31/4545;A61K31/496;A61K31/5377;A61K31/64;A61K38/28;A61K45/06;A61P3/04;A61P3/10;C07D249/08;C07D249/14;C07D401/04;C07D401/10;C07D401/12;C07D401/14;C07D403/04;C07D403/10;C07D405/04;C07D409/04;C07D413/10;C07D491/10 |
主分类号 |
A61K31/4196 |
代理机构 |
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代理人 |
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地址 |
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