发明名称 |
PIPECOLIC LINKER AND ITS USE FOR CHEMISTRY ON SOLID SUPPORT |
摘要 |
<p>The present invention relates to a pipecolic linker and its use as a solid-phase linker in organic synthesis. Said pipecolic solid-phase linker may be used for coupling functional groups chosen between primary amines, secondary amines, aromatic amines, alcohols, phenols and thiols. In particular, said pipecolic solid-phase linker may be used for peptide or pseudopeptide synthesis, such as the reverse N to C peptide synthesis or the retro-inverso peptide synthesis, or for the synthesis of small organic molecules.</p> |
申请公布号 |
WO2010023295(A1) |
申请公布日期 |
2010.03.04 |
申请号 |
WO2009EP61171 |
申请日期 |
2009.08.28 |
申请人 |
CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS);UNIVERSITE DE MONTPELLIER I;MARTINEZ, JEAN;ZAJDEL, PAWEL;PAWLOWSKI, MACIEJ;SUBRA, GILLES |
发明人 |
MARTINEZ, JEAN;ZAJDEL, PAWEL;PAWLOWSKI, MACIEJ;SUBRA, GILLES |
分类号 |
C07D211/60;C07B61/00;C08F8/10 |
主分类号 |
C07D211/60 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|