发明名称 Process for the preparation of [(1R), 2S]-2-aminopropionic acid 2-[4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-methylpyrrolo[2, 1-F][1,2,4]triazin-6-yloxy]-1-methylethyl ester
摘要 The invention relates to an improved process for preparing [(1R), 2S]-2-aminopropionic acid 2-[4-(4-fluoro-2-methyl-1H-indol-5-yloxy)-5-methylpyrrolo[2,1-f][1,2,4]triazin-6-yloxy]-1-methylethyl ester of the formula: Compound I has been shown to be useful for the treatment of certain types of cancer.
申请公布号 US7671199(B2) 申请公布日期 2010.03.02
申请号 US20070737787 申请日期 2007.04.20
申请人 BRITSOL-MYERS SQUIBB COMPANY 发明人 CRISPINO GERARD A.;HAMEDI MOURAD;LAPORTE THOMAS L.;THORNTON JOHN E.;PESTI JAAN A.;XU ZHONGMIN;LOBBEN PAUL C.;LEAHY DAVID K.;MUSLEHIDDINOGLU JALE;LAI CHIAJEN;SPANGLER LORI ANN;DISCORDIA ROBERT P.;GIBSON FRANCIS S.
分类号 C07D487/04;A61K31/53;A61P3/10 主分类号 C07D487/04
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