New substituted indole-carboxamide compounds useful e.g. in plant protection, for combating animal pests, arthropods, nematodes and plant diseases, and for protecting industrial materials against attack and destruction by insects

摘要

Substituted indole-carboxamide compounds (I) and their salts and N-oxides are new. Substituted indole-carboxamide compounds of formula (I) and their salts and N-oxides are new. X : O or S; A 1>, A 2>N or C-Y 1>, where A 1>, A 2>are not N at the same time; either R 1>1-8C alkyl, 3-7C cycloalkyl, 1-8C alkylcarbonyl, 1-8C alkoxycarbonyl, 2-8C alkenyl, 3-8C alkylalkenyl, 1-8C haloalkyl, phenylcarbonyl or benzyl (all optionally substituted) or H; and R 2>1-8C alkyl, aryl, benzyl, 3-7C cycloalkyl, 2-8C alkoxyalkyl or 1-8C haloalkyl (all optionally substituted); or R 1>R 2>5- or 6-membered ring (optionally substituted); either R 3>1-8C alkyl, aryl, 1-8C haloalkyl, 2-8C alkoxyalkyl or benzyl (all optionally substituted); and Y 1>H, NH 2, OH, halo, nitro, cyano, isocyano, mercapto, isothiocyanato, carboxy, carboxamide, SF 5, aminosulfonyl, 1-8C alkyl, 3-7C cycloalkyl, 2-8C alkenyl, 3-7C cycloalkyl, 2-8C alkynyl, N-mono-(1-8C)-alkylamino, N,N-di(1-8C)-alkylamino, N-(1-8C)-alkanoylamino, 1-8C alkoxy, 2-8C alkenyloxy, 2-8C alkynyloxy, 3-7C cycloalkoxy, 3-7C cycloalkenyloxy, 1-8C alkoxycarbonyl , 2-8C alkenyloxycarbonyl, 2-8C alkynyloxycarbonyl, aryloxycarbonyl, 1-8C alkanoyl, 2-8C alkenylcarbonyl, 2-8C alkynylcarbonyl, arylcarbonyl, 1-8C alkylthio, 3-7C cycloalkylthio, 2-8C alkenylthio, 3-7C cycloalkenylthio, 2-8c alkynylthio, 1-8C alkylsulfenyl or 1-8C alkylsulfinyl (where both enantiomers of alkylsulfinyl group are included), 1-8C alkylsulfonyl, N-mono(1-8C)-alkylamino-sulfonyl, N,N-di(1-8C)-alkylaminosulfonyl, 1-8C alkylphosphinyl, 1-8C alkylphosphonyl (where for alkylphosphinyl or alkylphosphonyl both enantiomers are included), N-(1-8C)-alkylaminocarbonyl, N,N-di(1-8C)-alkylaminocarbonyl, N-(1-8C)-alkanoylamino-carbonyl, N-(1-8C)-alkanoyl-N-(1-8C)-alkylaminocarbonyl, aryl, aryloxy, benzyl, benzyloxy, benzylthio, arylthio, arylamino, benzylamino, (2-7C)-heterocyclyl, tri(1-8C)-alkylsilyl, 1-8C alkoxy(1-8C) alkyl, 1-8C alkylthio(1-8C)-alkyl, 1-8C alkylthio (1-8C)-alkoxy, 1-8C alkoxy(1-8C)-alkoxy, phenethyl, benzyloxy, 1-8C haloalkyl, 3-7C halocycloalkyl, 1-8C alkyl, 1-8C haloalkylthio, 1-8C haloalkylsulfinyl, 1-8C haloalkylsulfonyl, 1-8C haloalkanoyl, 1-8C haloalkylcarbonyl, 2-8C haloalkoxy-carbonyl, halo(1-8C)-alkoxy(1-8C)-alkoxy, halo(1-8C)-alkoxy(1-8C)-alkylthio, halo(1-8C)alkoxy(1-8C)-alkanoyl or halo(1-8C)-alkoxy(1-8C)-alkyl; or R 3>Y 1>5- or 6-membered ring (optionally substituted); and m : 1-4. [Image] ACTIVITY : Plant Protectant; Arthropodicide; Nematocide; Insecticide; Antifouling; Arachnicide; Acaricide; Antiparasitic; Antihelmintic; Protozoacide. MECHANISM OF ACTION : None given.