发明名称 DIAZEPAN AND PIPERAZINE DERIVATIVES MODULATORS OF CHEMOKINE RECEPTORS
摘要 <p>The invention is concerned with novel heterocyclyl compounds of formula (I) wherein A, X, R3, R4, R5, R6, R7, R8, R9, R10, m, n and p are as defined in the description and in the claims, as well as physiologically acceptable salts thereof. These compounds are antagonists of CCR2 receptor, CCR5 receptor and/or CCR3 receptor and can be used as medicaments.</p>
申请公布号 WO2010012619(A1) 申请公布日期 2010.02.04
申请号 WO2009EP59270 申请日期 2009.07.20
申请人 F. HOFFMANN-LA ROCHE AG;ADAM, JEAN-MICHEL;AEBI, JOHANNES;BINGGELI, ALFRED;GREEN, LUKE;HARTMANN, GUIDO;MAERKI, HANS, P.;MATTEI, PATRIZIO;RICKLIN, FABIENNE;ROCHE, OLIVIER 发明人 ADAM, JEAN-MICHEL;AEBI, JOHANNES;BINGGELI, ALFRED;GREEN, LUKE;HARTMANN, GUIDO;MAERKI, HANS, P.;MATTEI, PATRIZIO;RICKLIN, FABIENNE;ROCHE, OLIVIER
分类号 C07D241/08;A61K31/4965;A61K31/551;A61P9/00;A61P29/00;C07D243/08;C07D401/06;C07D401/14;C07D413/06 主分类号 C07D241/08
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