发明名称 AMORPHOUS SUBSTANCE OF TRICYCLIC TRIAZOLOBENZAZEPINE DERIVATIVE
摘要 Disclosed are 2-(1-isopropoxycarbonyloxy-2-methylpropyl)-7,8-dimethoxy-4(5H),10-dioxo-2H-1,2,3-triazolo[4,5-c][1]benzazepine, which has been rendered amorphous and possesses improved absorption and dissoluvability, and a pharmaceutical composition comprising the same. Also disclosed are processes for producing 2-(1-isopropoxycarbonyloxy-2-methylpropyl)-7,8-dimethoxy-4(5H),10-dioxo-2H-1,2,3-triazolo[4,5-c][1]benzazepine, which has been rendered amorphous, and a pharmaceutical composition comprising the same.
申请公布号 CA2471651(C) 申请公布日期 2010.01.26
申请号 CA20022471651 申请日期 2002.12.25
申请人 MEIJI SEIKA KAISHA, LTD. 发明人 ISHIKURA, TOYOAKI;ISHIZAWA, TAKAYUKI;SUEMUNE, KENJI;ISHIWATA, MAYUMI;UDAGAWA, CHIKAKO
分类号 C07D487/04;A61K9/14;A61K31/55;A61K47/38;A61P29/00;A61P37/08 主分类号 C07D487/04
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