发明名称 |
METHOD FOR PRODUCING INTERMEDIATES FOR THE PRODUCTION OF NOVEL MACROCYCLES THAT ARE INHIBITORS OF THE PROTEASOMIC DEGRADATION OF P27, SUCH AS ARGYRIN AND DERIVATIVES THEREOF, AND USES OF SAID MACROCYCLES |
摘要 |
The present invention relates to the use of particular macrocycles that are inhibitors of the proteasomic degradation of p27, in particular argyrin and derivatives thereof, for a treatment in a variety of conditions, such as the induction of immunotolerance, autoimmune diseases, bacterial infections, and proliferative diseases, such as cancers. |
申请公布号 |
CA2729188(A1) |
申请公布日期 |
2010.01.21 |
申请号 |
CA20092729188 |
申请日期 |
2009.06.23 |
申请人 |
HELMHOLTZ-ZENTRUM FUER INFEKTIONS-FORSCHUNG GMBH;MEDIZINISCHE HOCHSCHULE HANNOVER;GOTTFRIED WILHELM LEIBNIZ UNIVERSITAET HANNOVER |
发明人 |
KALESSE, MARKUS;MALEK, NISAR;FRANK, RONALD;BRODMANN, TOBIAS;BUELOW, LEILA;RENTSCH, ANDREAS;GIRBIG, ANNA-KATHARINA;EGGERT, ULRIKE |
分类号 |
C07K7/56;A61K38/04 |
主分类号 |
C07K7/56 |
代理机构 |
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代理人 |
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地址 |
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