发明名称 Process for the preparation of (R)-(+)-4-(Ethylamino)-3,4-dihydro-2-(3-methoxypropyl)-2H-thieno[3,2-e]-1,2-thiazine-6-sulfonamide-1,1-dioxide.
摘要 Disclosed herein is an improved process for the preparation of (R)-(+)-4-(Ethylamino)-3,4-dihydro-2-(3-methoxypropyl)-2H-thieno[3,2-e]-1,2-thiazine-6-sulfonamide-1,1-dioxide (Brinzolamide) and novel intermediates thereof.
申请公布号 US2010009977(A1) 申请公布日期 2010.01.14
申请号 US20070443836 申请日期 2007.10.12
申请人 SATHE DHANANJAY GOVIND;TARUR RADHAKRISHNAN VENKATASUB;BHISE NANDU BABAN;SHINDE AJIT BHASKAR;PARDESHI SANTOSH 发明人 SATHE DHANANJAY GOVIND;TARUR RADHAKRISHNAN VENKATASUBRAMANIAN;BHISE NANDU BABAN;SHINDE AJIT BHASKAR;PARDESHI SANTOSH
分类号 A61K31/54;A61P9/12;C07D513/04 主分类号 A61K31/54
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