发明名称 |
Process for the preparation of (R)-(+)-4-(Ethylamino)-3,4-dihydro-2-(3-methoxypropyl)-2H-thieno[3,2-e]-1,2-thiazine-6-sulfonamide-1,1-dioxide. |
摘要 |
Disclosed herein is an improved process for the preparation of (R)-(+)-4-(Ethylamino)-3,4-dihydro-2-(3-methoxypropyl)-2H-thieno[3,2-e]-1,2-thiazine-6-sulfonamide-1,1-dioxide (Brinzolamide) and novel intermediates thereof.
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申请公布号 |
US2010009977(A1) |
申请公布日期 |
2010.01.14 |
申请号 |
US20070443836 |
申请日期 |
2007.10.12 |
申请人 |
SATHE DHANANJAY GOVIND;TARUR RADHAKRISHNAN VENKATASUB;BHISE NANDU BABAN;SHINDE AJIT BHASKAR;PARDESHI SANTOSH |
发明人 |
SATHE DHANANJAY GOVIND;TARUR RADHAKRISHNAN VENKATASUBRAMANIAN;BHISE NANDU BABAN;SHINDE AJIT BHASKAR;PARDESHI SANTOSH |
分类号 |
A61K31/54;A61P9/12;C07D513/04 |
主分类号 |
A61K31/54 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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