发明名称 CRYSTALLINE FORMS OF ERLOTINIB BASE AND ERLOTINIB HCL
摘要 The preparation of crystalline Erlotinib base form G2 is described. This crystalline form can be converted to an Erlotinib salt, such as Erlotinib HCl, which can be used in the treatment of patients with locally advanced or metastatic non-small cell lung cancer (NSCLC).
申请公布号 US2010004449(A1) 申请公布日期 2010.01.07
申请号 US20090498543 申请日期 2009.07.07
申请人 PLUS CHEMICALS SA 发明人 GAVENDA ALES;VRASPIR PAVEL;CANAVESI AUGUSTO;ARONHIME JUDITH;BIGATTI ETTORE;FAUSTMANN JIRI;JEGOROV ALEXANDR;STEPHENS PETER W.;LUX GIOVANNA;PAIOCCHI MAURIZIO
分类号 C07D239/72 主分类号 C07D239/72
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