PROCESS FOR THE PREPARATION OF BENZOIMIDAZOL-2-YL PYRIMIDINE DERIVATIVES
摘要
The present invention is directed to processes for the preparation of benzoimidazol-2-yl pyrimidine derivatives useful as histamine H4 receptor modulators, and a crystalline hemi-tartrate of [5-(4,6-dimethyl-1H-benzoimidazol-2-yl)-4-methyl-pyrimidin-2-yl]-[3-(1-methyl-piperidin-4-yl)-propyl]-amine.
申请公布号
CA2729703(A1)
申请公布日期
2010.01.07
申请号
CA20092729703
申请日期
2009.06.29
申请人
JANSSEN PHARMACEUTICA NV
发明人
CESCO-CANCIAN, SERGIO;GRIMM, JEFFREY S.;MANI, NEELAKANDHA S.;MAPES, CHRISTOPHER M.;PALMER, DAVID C.;PIPPEL, DANIEL J.;XIAO, TONG;BROGGINI, DIEGO;LOCHNER, SUSANNE