发明名称 PROCESS FOR THE PREPARATION OF BENZOIMIDAZOL-2-YL PYRIMIDINE DERIVATIVES
摘要 The present invention is directed to processes for the preparation of benzoimidazol-2-yl pyrimidine derivatives useful as histamine H4 receptor modulators, and a crystalline hemi-tartrate of [5-(4,6-dimethyl-1H-benzoimidazol-2-yl)-4-methyl-pyrimidin-2-yl]-[3-(1-methyl-piperidin-4-yl)-propyl]-amine.
申请公布号 CA2729703(A1) 申请公布日期 2010.01.07
申请号 CA20092729703 申请日期 2009.06.29
申请人 JANSSEN PHARMACEUTICA NV 发明人 CESCO-CANCIAN, SERGIO;GRIMM, JEFFREY S.;MANI, NEELAKANDHA S.;MAPES, CHRISTOPHER M.;PALMER, DAVID C.;PIPPEL, DANIEL J.;XIAO, TONG;BROGGINI, DIEGO;LOCHNER, SUSANNE
分类号 C07D403/04;A61K31/506 主分类号 C07D403/04
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