发明名称 CRYSTALLINE FORMS OF ((((4-((5-(CYCLOPROPYLCARBAMOYL)-2-METHYLPHENYL)AMINO)-5-METHYLPYRROLO[2,1-F][1,2,4]TRIAZIN-6-YL)CARBONYL)(PROPYL)CARBAMOYL)OXY)METHYL (4-(PHOSPHONOOXY)PHENYL)ACETATE, PREPARATION AND USE THEREOF
摘要 <p>The present invention generally relates to crystalline forms of ((((4-((5- (cyclopropylcart&gt;amoyl)-2-methylphenyl)amino)-5-methylpyrrolo[2, 1 -J][ I,2,4]triazin- 6-yl)carbonyl)(propyl)carbamoyl)oxy)methyl (4-(phosphonooxy)phenyl)acetate. The present invention also generally relates to a pharmaceutical composition comprising said crystalline form, as well of methods of obtaining and using the crystalline form for the treatment of inflammatory-associated diseases.</p>
申请公布号 WO2009158450(A1) 申请公布日期 2009.12.30
申请号 WO2009US48560 申请日期 2009.06.25
申请人 BRISTOL-MYERS SQUIBB COMPANY;MALLEY, MARY, F.;DIMARCO, JOHN, D.;GALELLA, MICHAEL;GOUGOUTAS, JACK, Z.;YIN, XIAOTIAN, S. 发明人 MALLEY, MARY, F.;DIMARCO, JOHN, D.;GALELLA, MICHAEL;GOUGOUTAS, JACK, Z.;YIN, XIAOTIAN, S.
分类号 C07F9/6561 主分类号 C07F9/6561
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