发明名称 FUSED HETEROCYCLES
摘要 This invention provides fused heterocycles having the formula: in which R1 is a member selected from the group consisting of H, substituted or unsubstituted arylalkyl and substituted or unsubstituted heteroarylalkyl. R2 is a member selected from the group consisting of H substituted or unsubstituted alkenyl, substituted or unsubstituted arylalkyl and substituted or unsubstituted heteroarylalkyl. R3 is a member selected from the group consisting of H1 C1-C6 substituted or unsubstituted alkyl, substituted or unsubstituted arylalkyl and substituted or unsubstituted heteroarylalkyl. R4 is a member selected from OH and O- X+, in which X+ is positive ion which is a member selected from organic positive ions and inorganic positive ions. Substituted or unsubstituted arylalkyl and substituted or unsubstituted heteroarylalkyl moieties have the formula: in which Ar is a member selected from the group consisting of substituted or unsubstituted aryl and substituted or unsubstituted heteroaryl. The index n is an integer from 1 to 4. Formulae A, B.
申请公布号 WO2009020814(A3) 申请公布日期 2009.12.30
申请号 WO2008US71642 申请日期 2008.07.30
申请人 SEPRACOR INC.;HEFFERNAN, MICHELE, L.R.;DORSEY, JAMES, M.;FANG, QUN, KEVIN;FOGLESONG, ROBERT, J.;HOPKINS, SETH, C.;OGBU, CYPRIAN, O.;SOUKRI, MUSTAPHA;SPEAR, KERRY, L. 发明人 HEFFERNAN, MICHELE, L.R.;DORSEY, JAMES, M.;FANG, QUN, KEVIN;FOGLESONG, ROBERT, J.;HOPKINS, SETH, C.;OGBU, CYPRIAN, O.;SOUKRI, MUSTAPHA;SPEAR, KERRY, L.
分类号 A01N43/16;A61K31/35 主分类号 A01N43/16
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