发明名称 INDOLYLMALEIMIDE DERIVATIVES AS PROTEIN KINASE C INHIBITORS
摘要 The invention provides indolylmaleimide derivatives of formula I (see formula I) The derivatives may be used to treat or prevent T-cell mediated acute or chronic inflammatory diseases or disorders, autoimmune diseases, graft rejection or cancer.
申请公布号 CA2428133(C) 申请公布日期 2009.12.29
申请号 CA20012428133 申请日期 2001.11.05
申请人 NOVARTIS AG 发明人 COOKE, NIGEL GRAHAM;COTTENS, SYLVAIN;EHRHARDT, CLAUS;VON MATT, PETER;SEDRANI, RICHARD;WAGNER, JURGEN;EVENOU, JEAN-PIERRE;ALBERT, RAINER;ZENKE, GERHARD
分类号 C07D403/14;A61K31/404;A61K31/4178;A61K31/4439;A61K31/454;A61K31/496;A61K31/506;A61K31/517;A61K31/527;A61K31/5377;A61K31/551;A61K45/06;A61P1/04;A61P1/16;A61P3/02;A61P3/10;A61P5/14;A61P9/00;A61P9/04;A61P9/10;A61P9/12;A61P11/00;A61P11/06;A61P13/12;A61P17/00;A61P17/06;A61P19/02;A61P21/00;A61P21/04;A61P25/00;A61P25/28;A61P27/02;A61P29/00;A61P31/18;A61P35/00;A61P37/02;A61P37/04;A61P37/06;A61P37/08;A61P43/00;C07D401/14;C07D403/04;C07D471/10;C07D521/00 主分类号 C07D403/14
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