发明名称 |
PROCESSES FOR THE PREPARATION OF STATINS, PARTICULARLY ROSUVASTATIN, AND INTERMEDIATES FOR THE PREPARATION THEREOF |
摘要 |
The process for the synthesis of statins featuring the use of an early intermediate (4R,6S)-6-(dialkoxymethyl)tetrahydro-2H-pyran-2,4-diol which already possesses the desired stereochemistry corresponding to the final statin. |
申请公布号 |
EP2134696(A2) |
申请公布日期 |
2009.12.23 |
申请号 |
EP20080718383 |
申请日期 |
2008.04.02 |
申请人 |
LEK PHARMACEUTICALS D.D. |
发明人 |
CASAR, ZDENKO;MESAR, TOMAZ;KOPITAR, GREGOR;MRAK, PETER;OSLAJ, MATEJ |
分类号 |
C07D239/42;A61K31/506;C07D309/30;C07H3/02 |
主分类号 |
C07D239/42 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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