发明名称 PROCESSES FOR THE PREPARATION OF STATINS, PARTICULARLY ROSUVASTATIN, AND INTERMEDIATES FOR THE PREPARATION THEREOF
摘要 The process for the synthesis of statins featuring the use of an early intermediate (4R,6S)-6-(dialkoxymethyl)tetrahydro-2H-pyran-2,4-diol which already possesses the desired stereochemistry corresponding to the final statin.
申请公布号 EP2134696(A2) 申请公布日期 2009.12.23
申请号 EP20080718383 申请日期 2008.04.02
申请人 LEK PHARMACEUTICALS D.D. 发明人 CASAR, ZDENKO;MESAR, TOMAZ;KOPITAR, GREGOR;MRAK, PETER;OSLAJ, MATEJ
分类号 C07D239/42;A61K31/506;C07D309/30;C07H3/02 主分类号 C07D239/42
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