发明名称 A POLYMORPHIC FORM OF A PYRAZINO [2, 3-H] [3] BENZAZEPINE DERIVATIVE
摘要 The invention relates generally to a crystalline polymorphic form of 7, 8, 9, 10-tetrahydro-6, 10-methano-6H-pyrazino[2, 3-h][3] benzazepine, varenicline base, i.e. a hydrate of varenicline base, designated herein as Form II, and to a method for preparing and obtaining the same.
申请公布号 WO2009101185(A3) 申请公布日期 2009.12.03
申请号 WO2009EP51727 申请日期 2009.02.13
申请人 MEDICHEM, S.A.;WINTER, STEPHEN, BENEDICT, DAVID 发明人 WINTER, STEPHEN, BENEDICT, DAVID
分类号 C07D471/08;A61P25/34 主分类号 C07D471/08
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