PROCESS FOR THE GLYCOSIDATION OF COLCHICINE AND THIOCOLCHICINE
摘要
<p>A process for the preparation of compounds having formula (I) is disclosed, wherein: - R1 is a methoxy or methylthio group; - R2 is a O-glycosyloxy residue. Compounds having formula (I) are prepared by reacting the corresponding precursor having R2 = OH and the suitably protected 1-acetyl- glycose.</p>