摘要 |
A NOVEL COMPOUND OF THE FORMULA (I): WHEREIN RI IS ALKOXYCARBONYL OR THE LIKE, R2 IS ALKYL OR THE LIKE; R3 IS HYDROGEN OR THE LIKE; R4 IS ALKYLENE OR THE LIKE; R5 IS OPTIONALLY SUBSTITUTED HETEROCYCLIC GROUP; R6, R7, AND R8 ARE INDEPENDENTLY HYDROGEN; ALKYL, ALKOXY, OR THE LIKE; RIO IS OPTIONALLY SUBSTITUTED AROMATIC RING, OR THE LIKE; OR A PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, WHICH HAS AN INHIBITORY ACTIVITY AGAINST CHOLESTERYL ESTER TRANSFER PROTEIN (CETP).
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