发明名称 QUINUCLIDINE DERIVATIVES AND THEIR USE AS MUSCARINIC RECEPTOR ANTAGONISTS FOR THE TREATMENT OF ASTHMA AND CHRONIC OBSTRUCTIVE PULMONARY DISEASE (COPD)
摘要 <p>The invention provides compounds of formula (I) wherein R1, R2, R3, R4, R5, Het1, n, Y and X are as defined in the specification, a process for their preparation, pharmaceutical compositions containing them, a process for preparing pharmaceutical compositions, their use in therapy and intermediates of use in their preparation.</p>
申请公布号 WO2009139709(A1) 申请公布日期 2009.11.19
申请号 WO2009SE50526 申请日期 2009.05.12
申请人 ASTRAZENECA AB;ARGENTA DISCOVERY LTD.;FORD, RHONAN;MATHER, ANDREW;METE, ANTONIO;MILLICHIP, IAN 发明人 MATHER, ANDREW;METE, ANTONIO;MILLICHIP, IAN
分类号 C07D453/02;A61K31/439;A61P11/06;A61P11/08 主分类号 C07D453/02
代理机构 代理人
主权项
地址