发明名称 |
AN IMPROVED PROCESS FOR THE PREPARATION OF SOLIFENACIN AND ITS PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF |
摘要 |
The present invention relates to an improved process for the preparation of solifenacin compound of formula (1) and its succinate salt compound of formula (1a), comprising the condensation of (R)-3- quinuclidinol with (S)-ethyl- 1 -phenyl- 1,2,3,4-tetrahydro-2-isoquinoline carboxylate in presence of a suitable hydroxide base in a suitable solvent. |
申请公布号 |
WO2009139002(A2) |
申请公布日期 |
2009.11.19 |
申请号 |
WO2009IN00278 |
申请日期 |
2009.05.11 |
申请人 |
MSN LABORATORIES LIMITED;SATYANARAYANA REDDY, MANNE;ESWARAIAH, SAJJA;VENKATESH, MUMMADI |
发明人 |
SATYANARAYANA REDDY, MANNE;ESWARAIAH, SAJJA;VENKATESH, MUMMADI |
分类号 |
C07D453/02 |
主分类号 |
C07D453/02 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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