发明名称 SUNITINIB HEMI-L-MALATE, POLYMORPHS AND PREPARATION THEREOF, POLYMORPHS OF RACEMIC SUNITINIB MALATE, COMPOSITINS CONTAINING SUNITINIB BASE AND MALIC ACID AND PREPARATION THEREOF
摘要 The invention provides Sunitinib hemi-L-malate, polymorphs thereof, polymorphs of racemic sunitinib malate, compositions containing sunitinib base and either L or racemic malic acid, processes for the preparation thereof, and pharmaceutical compositions thereof.
申请公布号 WO2009067686(A3) 申请公布日期 2009.11.12
申请号 WO2008US84386 申请日期 2008.11.21
申请人 TEVA PHARMACEUTICAL INDUSTRIES LTD.;TEVA PHARMACEUTICALS USA, INC.;JEGOROV, ALEXANDR;GAVENDA, ALES;VRASPIR, PAVEL;ARONHIME, JUDITH;ANGIOLETTI, PAOLO;CANAVESI, AUGUSTO;VILLA, MARCO;SCARPITTA, FRANCESCA;BIGATTI, ETTORE;MACDONALD, PETER, LINDSAY 发明人 JEGOROV, ALEXANDR;GAVENDA, ALES;VRASPIR, PAVEL;ARONHIME, JUDITH;ANGIOLETTI, PAOLO;CANAVESI, AUGUSTO;VILLA, MARCO;SCARPITTA, FRANCESCA;BIGATTI, ETTORE;MACDONALD, PETER, LINDSAY
分类号 C07D403/06;A61K31/404;A61P35/00 主分类号 C07D403/06
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