发明名称 |
HETEROCYCLIC DERIVATIVES AS GPCR RECEPTOR AGONISTS |
摘要 |
Compounds of Formula (I), R1-A-V-B-R2; or pharmaceutically acceptable salts thereof, are agonists of GPR116 and are useful as regulators of satiety, e.g. for the treatment of obesity, and for the treatment of diabetes.
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申请公布号 |
US2009281060(A1) |
申请公布日期 |
2009.11.12 |
申请号 |
US20040584025 |
申请日期 |
2004.12.23 |
申请人 |
PROSIDION LIMITED |
发明人 |
FYFE MATTHEW;KING-UNDERWOOD JOHN;BERTRAM (GARDNER) LISA SARAH;THOMAS GERARD HUGH;PROCTER MARTIN;RASAMISON CHRYSTELLE;SCHOFIELD KAREN |
分类号 |
A61K31/4545;A61K31/454;A61K31/497;A61K31/675;A61P3/00;C07D401/14;C07D413/04;C07D413/06;C07D413/12;C07D413/14;C07D417/04;C07D417/14;C07F9/58 |
主分类号 |
A61K31/4545 |
代理机构 |
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主权项 |
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地址 |
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