发明名称 HETEROCYCLIC DERIVATIVES AS GPCR RECEPTOR AGONISTS
摘要 Compounds of Formula (I), R1-A-V-B-R2; or pharmaceutically acceptable salts thereof, are agonists of GPR116 and are useful as regulators of satiety, e.g. for the treatment of obesity, and for the treatment of diabetes.
申请公布号 US2009281060(A1) 申请公布日期 2009.11.12
申请号 US20040584025 申请日期 2004.12.23
申请人 PROSIDION LIMITED 发明人 FYFE MATTHEW;KING-UNDERWOOD JOHN;BERTRAM (GARDNER) LISA SARAH;THOMAS GERARD HUGH;PROCTER MARTIN;RASAMISON CHRYSTELLE;SCHOFIELD KAREN
分类号 A61K31/4545;A61K31/454;A61K31/497;A61K31/675;A61P3/00;C07D401/14;C07D413/04;C07D413/06;C07D413/12;C07D413/14;C07D417/04;C07D417/14;C07F9/58 主分类号 A61K31/4545
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