发明名称 SUBSTITUTED 8-PIPERIDINYL-2-PYRIDINYL-PYRIMIDO[1,2-a] PYRIMIDIN-6-ONE AND 8-PIPERIDINYL-2-PYRIMIDINYL-PYRIMIDO[1,2-a] PYRIMIDIN-6-ONE DERIVATIVES
摘要 The invention relates to a pyrimidone derivative represented by formula (I) or a salt thereof: Wherein X, Y, R1, R2, R3, R4, n, p, q, o and m are as described herein. The invention relates also to a medicament comprising the said derivative or a salt thereof as an active ingredient which is used for preventive and/or therapeutic treatment of a neurodegenerative disease caused by abnormal activity of GSK3beta, such as Alzheimer disease.
申请公布号 US2009281121(A1) 申请公布日期 2009.11.12
申请号 US20090434053 申请日期 2009.05.01
申请人 SANOFI-AVENTIS;MITSUBISHI TANABE PHARMA CORPORATION 发明人 LOCHEAD ALISTAIR;SAADY MOURAD;SLOWINSKI FRANCK;YAICHE PHILIPPE
分类号 A61K31/519;A61P3/00;A61P25/00;C07D487/04 主分类号 A61K31/519
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