发明名称 METHOD FOR SEMISYNTHESIS OF DESERPIDINE
摘要 FIELD: chemistry. ^ SUBSTANCE: invention relates to an improved highly-selective method of producing deserpidine (Ia) through demethylation of 11-methoxy group of 11-O-methyl reserpic acid lactone, with subsequent stages for reduction, hydrolysis and esterification of the obtained methyldeserpidate 3,4,5-trimethoxybenzoic acid. Output is 40%. ^ EFFECT: method for semisynthesis of deserpidine is described. ^ 6 cl, 7 ex
申请公布号 RU2372351(C2) 申请公布日期 2009.11.10
申请号 RU20060133740 申请日期 2005.03.02
申请人 INDENA S.P.A. 发明人 FONTANA GABRIELE;BOMBARDELLI EHTSIO;SAMORI KRISTIAN;BAL'DELLI EHLEONORA;GUERRINI ANDREA;BATTAL'JA ARTURO;DANIELI BRUNO
分类号 C07D459/00 主分类号 C07D459/00
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