发明名称 QUINOLINE OR ISOQUINOLINE SUBSTITUTED P2X7 ANTAGONISTS
摘要 <p>The present invention is related to novel compounds of formula (I) having P2X7 antagonistic properties, pharmaceutical compositions comprising these compounds, chemical processes for preparing these compounds and their use in the treatment or prophylaxis of diseases associated with P2X7 receptor activity in animals, in particular humans. (I)</p>
申请公布号 WO2009132000(A1) 申请公布日期 2009.10.29
申请号 WO2009US41249 申请日期 2009.04.21
申请人 JANSSEN PHARMACEUTICA NV;LOVE, CHRISTOPHER, JOHN;LEENAERTS, JOSEPH, ELISABETH;COOYMANS, LUDWIG, PAUL;LEBSACK, ALEC, DONALD;BRANSTETTER, BRYAN, JAMES;RECH, JASON, CHRISTOPHER;GLEASON, ELIZABETH, ANN;VENABLE, JENNIFER, DIANE;WIENER, DANIELLE;SMITH, DEBORAH, MARGARET;BREITENBUCHER, JAMES, GUY 发明人 LOVE, CHRISTOPHER, JOHN;LEENAERTS, JOSEPH, ELISABETH;COOYMANS, LUDWIG, PAUL;LEBSACK, ALEC, DONALD;BRANSTETTER, BRYAN, JAMES;RECH, JASON, CHRISTOPHER;GLEASON, ELIZABETH, ANN;VENABLE, JENNIFER, DIANE;WIENER, DANIELLE;SMITH, DEBORAH, MARGARET;BREITENBUCHER, JAMES, GUY
分类号 C07D401/14;A61K31/4427;C07D405/14;C07D413/14 主分类号 C07D401/14
代理机构 代理人
主权项
地址