发明名称 Fused heterocyclic derivative, medicinal composition containing the same, and medicinal use thereof
摘要 Provided is a compound useful as a preventive or therapeutic agent for sexual-hormone-dependent diseases, etc. It is a fused heterocyclic derivative represented by the following general formula (I). In the formula (I), ring A is a five-membered cyclic unsaturated hydrocarbon or five-membered heteroaryl; R<A> is halogeno, alkyl, alkenyl, alkynyl, carboxy, alkoxy, carbamoyl, alkylcarbamoyl, etc.; ring B is aryl or heteroaryl; R is halogeno, alkyl, carboxy, alkoxy, carbamoyl, alkylcarbamoyl, etc.; E<1> and E<2> each is oxygen, etc.; U is a single bond or alkylene; and X is, e.g., a group represented by Y, -SO2-Y, -O-(alkylene)-Y-, or -O-Z (wherein Y is Z, amino, etc. and Z is cycloalkyl, heterocycloalkyl, aryl, heteroaryl, etc.).
申请公布号 ZA200803335(B) 申请公布日期 2009.10.28
申请号 ZA20080003335 申请日期 2006.10.17
申请人 KISSEI PHARMACEUTICAL CO., LTD 发明人 OHNO, KOHSUKE;MIYAGI, TAKASHI;OZAWA, TOMONAGA;FUSHIMI, NOBUHIKO
分类号 A61K;A61P;C07D 主分类号 A61K
代理机构 代理人
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