发明名称 |
A NEW PROCESS FOR THE MANUFACTURING OF THE COMPOUND 2-HYDROXY-3-[5-(MORPHOLIN-4-YLMETHYL)PYRIDIN-2-YL]1H-INDOLE-5-C ARBONITRILE 701. |
摘要 |
<p>The present invention relates to a new process for the manufacture of the compound 2-hydroxy-3-[5-(morpholin-4-ylmethyl)pyridin-2-yl]1H-ind ole-5-carbonitrile as a free base and pharmaceutically acceptable salts thereof, particularly the 2-hydroxy-3-[5-(morpholin-4-ylmethyl)pyridin-2-yl]1H-ind ole-5-carbonitrile citrate, and to new intermediates prepared in said process suitable for large scale manufacturing of said compound.</p> |
申请公布号 |
MX2009010890(A) |
申请公布日期 |
2009.10.26 |
申请号 |
MX20090010890 |
申请日期 |
2008.04.17 |
申请人 |
ASTRAZENECA AB |
发明人 |
MARTIN HEDBERG;VERN DELISSER;ANNETTE JANSSON;ANDREAS RAADEVIK;PER RYBERG;SWANTJE THIERING |
分类号 |
C07D401/04;A61K31/5355;C07D213/38 |
主分类号 |
C07D401/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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