发明名称 |
INDOLES AS MODULATORS OF NICOTICIC ACETYLCHOLINE RECEPTOR SUBTYPE ALPHA-7 |
摘要 |
This invention relates to modulation of the a7 nicotinic acetylcholine receptor (nAChR) by a compound of List A or a salt thereof which may be represented by N-[(2-Trifluoromethyl-1H-indol-5-yl)methyl]-5-(trifluoromethyl)-2-pyrimidinecarboxarnide.
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申请公布号 |
CA2721630(A1) |
申请公布日期 |
2009.10.22 |
申请号 |
CA20092721630 |
申请日期 |
2009.04.16 |
申请人 |
GLAXO GROUP LIMITED |
发明人 |
DINNELL, KEVIN;LIGHTFOOT, ANDREW P.;MARSHALL, HOWARD ROBERT |
分类号 |
C07D401/12;A61K31/4439;A61P25/18 |
主分类号 |
C07D401/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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