发明名称 PROCESS AND INTERMEDIATES FOR THE SYNTHESIS OF 8-[{1-(3,5-BIS-(TRIFLUOROMETHYL)PHENYL)-ETHOXY}-METHYL]-8-PHENY L-1,7-DIAZA-SPIRO[4.5]DECAN-2-ONE COMPOUNDS.
摘要 <p>This application discloses a process to synthesize 8-({1-(3,5-Bis- (trifluoromethyl)phenyl)-ethoxy)-methyl]-8-pheny-1.7-diaza-sÏ¿i ro[4.5]decan-2-one comprising reacting a compound of the Formula 27a-sulfonate with zinc in the presence of acetic acid.</p>
申请公布号 MX2009010211(A) 申请公布日期 2009.10.19
申请号 MX20090010211 申请日期 2008.03.20
申请人 SCHERING CORPORATION. 发明人 PALIWAL, SUNIL;SHIH, NENG-YANG;MERGELSBERG, INGRID;SCHERER, DOMINIK HERMANN;HUTTENLOCH, MONIKA ERIKA;TSUI, HON-CHUNG
分类号 C07D211/38;C07D471/10;C07D498/10 主分类号 C07D211/38
代理机构 代理人
主权项
地址