发明名称 1H-Indole-Pyridinecarboxamide and 1H-Indole-Piperidinecarboxamide Compounds
摘要 Compounds of formula (I): wherein: A represents a divalent radical: wherein: Z represents an oxygen atom or a sulphur atom, R6 represents a hydrogen atom, an alkyl, alkenyl, arylalkyl or polyhaloalkyl group or a substituted, linear or branched alkyl chain, <img id="CUSTOM-CHARACTER-00001" he="1.78mm" wi="7.03mm" file="US20090258883A1-20091015-P00001.TIF" img-content="character" img-format="tif"/> represents a single bond or a double bond, R1, R2, R3 and R4 represent a hydrogen or halogen atom, an alkyl, alkoxy, hydroxy, cyano, nitro, polyhaloalkyl or optionally substituted amino group, or a linear or branched alkyl chain substituted by one or more groups, R5 represents a hydrogen atom or an alkyl, aminoalkyl or hydroxyalkyl group, X and Y represent a hydrogen atom or an alkyl group, Ra, Rb, Rc and Rd represent a hydrogen or halogen atom, an alkyl, hydroxy, alkoxy, cyano, nitro, polyhaloalkyl, optionally substituted amino group, or a substituted, linear or branched alkyl chain, Re represents a hydrogen atom or an alkyl, arylalkyl or alkenyl group or a substituted, linear or branched alkyl chain, their enantiomers, diastereoisomers, and N-oxides, and also addition salts thereof with a pharmaceutically acceptable acid or base.
申请公布号 US2009258883(A1) 申请公布日期 2009.10.15
申请号 US20060988424 申请日期 2006.07.06
申请人 LES LABORATOIRES SERVIER;CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE;UNIVERSITE PARIS SUD 发明人 BRION JEAN-DANIEL;BINTEIN FABRICE;RAZET RODOLPHE;RAZON PATRICK;RENKO ZAFIARISOA DOLOR;LEVOIRIER ERIC;PUJOL JEAN-FRANCOIS;WEISSMANN DINAH;LE RIDANT ALAIN;HARPEY CATHERINE
分类号 A61K31/496;A61K31/4439;A61K31/454;A61P25/16;A61P25/22;A61P25/24;A61P25/28;C07D401/12;C07D401/14 主分类号 A61K31/496
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