METHOD FOR THE ENZYMATIC KINETIC RESOLUTION OF ACYLOXYALKYL THIOCARBONATES USED FOR THE SYNTHESIS OF ACYLOXYALKYL CARBAMATES
摘要
<p>Methods of enzymatically resolving acyloxyalkyl thiocarbonates useful in the synthesis of acyloxyalkyl carbamates are disclosed. These carbamates can be coupled to drugs containing amines such as R-baclofen or S-pregabalin.</p>
申请公布号
WO2009094569(A3)
申请公布日期
2009.10.08
申请号
WO2009US31873
申请日期
2009.01.23
申请人
XENOPORT, INC.;GALLOP, MARK A.;YAO, FENMEI;LUDWIKOW, MARIA J.;PENG, GE;RAILLARD, STEVEN P.
发明人
GALLOP, MARK A.;YAO, FENMEI;LUDWIKOW, MARIA J.;PENG, GE;RAILLARD, STEVEN P.
