发明名称 |
NOVEL INTERMEDIATE FOR GLYT1 INHIBITOR |
摘要 |
This invention relates to an improved process for preparing the glycine transport 1 (GlyT1) inhibitor (Z)-N-(1-(4-(2-furyl)phenyl)-1-(3-thienyl-prop-1-en-3-yl) sarcosine via the novel intermediate (Z)-3-(4-(2-furyl)phenyl)-3-(3-thienyl)-prop-2-en-1-ol and the preparation of the latter.
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申请公布号 |
US2009253918(A1) |
申请公布日期 |
2009.10.08 |
申请号 |
US20070444010 |
申请日期 |
2007.09.26 |
申请人 |
JANSSEN PHARMACEUTICALS, N.V. |
发明人 |
HOUPIS IOANNIS NICOLAOS;SCHILS DIDIER PHILIPPE ROBERT |
分类号 |
C07D409/10 |
主分类号 |
C07D409/10 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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