发明名称 2H-BENZO[b][1,4]OXAZIN-3(4H)-ONE DERIVATIVES FOR USE AS STEAROYL CoA DESATURASE INHIBITORS
摘要 The present invention discloses 2H-benzo[b][1,4]oxazin-3(4H)-one derivatives for use as inhibitors of stearoyl-CoA desaturase having the structure of Formula I: The compounds are useful in treating and/or preventing various human diseases, mediated by stearoyl-CoA desaturase (SCD) enzymes, especially diseases related to abnormal lipid levels, cardiovascular disease, diabetes, obesity, metabolic syndrome and the like.
申请公布号 US2009253693(A1) 申请公布日期 2009.10.08
申请号 US20090417854 申请日期 2009.04.03
申请人 KOLTUN DMITRY;ZABLOCKI JEFF;VASILEVICH NATALYA;MIGULIN VASILY 发明人 KOLTUN DMITRY;ZABLOCKI JEFF;VASILEVICH NATALYA;MIGULIN VASILY
分类号 A61K31/538;A61P9/00;C07D265/36 主分类号 A61K31/538
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