| 发明名称 |
PRODRUGS OF PIPERAZINE AND SUBSTITUTED PIPERIDINE ANTIVIRAL AGENTS. |
| 摘要 |
THIS INVENTION PROVIDES FOR PRODRUG COMPOUNDS &Igr;, PHARMACEUTICAL COMPOSITIONS THEREOF, AND THEIR USE IN TREATING HIV INFECTION. WHEREIN: X IS C OR N WITH THE PROVISO THAT WHEN X IS N, R¹ DOES NOT EXIST; W IS C OR N WITH THE PROVISO THAT WHEN W IS N, R² DOES NOT EXIST; V IS C; E IS HYDROGEN OR A PHARMACEUTICALLY ACCEPTABLE SALT THEREOF; AND Y IS SELECTED FROM THE GROUP CONSISTING OF ALSO, THIS INVENTION PROVIDES FOR INTERMEDIATE COMPOUNDS &Igr;&Igr; USEFUL IN MAKING PRODRUG COMPOUNDS &Igr;. |
| 申请公布号 |
MY139243(A) |
申请公布日期 |
2009.09.30 |
| 申请号 |
MY2005PI01051 |
申请日期 |
2005.03.12 |
| 申请人 |
BRISTOL-MYERS SQUIBB COMPANY |
发明人 |
YASUTSUGU UEDA;SHAWN K. PACK;NACHIMUTHU SOUNDARARAJAN;PIERRE SIRARD;KATHIA LEVESQUE;DOMINIQUE THORAVAL;TIMOTHY P. CONNOLLY;JOHN F. KADOW;NICHOLAS A. MEANWELL;TAO WANG;CHUNG-PIN H. CHEN;KAP-SUN YEUNG;ZHONGXING ZHANG;DAVID KENNETH LEAHY |
| 分类号 |
A61K31/437;A61K31/496;A61K31/675;C07D471/04;C07F9/09;C07F9/572;C07F9/6561 |
主分类号 |
A61K31/437 |
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