发明名称 Pyridazine derivatives and their use as therapeutic agents
摘要 Compounds for treating an SCD-mediated disease or condition in a mammal, preferably a human, are disclosed, wherein the compounds are of formula (I): where x y, W, V, R 2 , R 3 , R 4 , R 5 , R 6 , R 6a , R 7 , R 7a , R 8 , R 8a , R 9 and R 9a are defined herein. Pharmaceutical compositions comprising the compounds of formula (I) are also disclosed.
申请公布号 AU2004261252(C1) 申请公布日期 2009.09.17
申请号 AU20040261252 申请日期 2004.07.29
申请人 XENON PHARMACEUTICALS INC. 发明人 VISHNUMURTHY KODUMURU;SENGEN SUN;NAGASREE CHAKKA;MARK W. HOLLADAY;MICHAEL D. WINTHER;VANDNA RAINA;SULTAN CHOWDHURY;SHIFENG LIU;SERGUEI SVIRIDOV;CHI TU;JIAN-MIN FU;DUANJIE HOU;MIKHAIL CHAFEEV;WENBAO LI;ZAIHUI ZHANG;RAJENDER KAMBOJ;HEINZ W. GSCHWEND;MELWYN ABREO;SHAOYI SUN
分类号 A61K31/00;A61K31/501;A61K31/551;A61P3/06;C07D237/20;C07D237/24 主分类号 A61K31/00
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