发明名称 AZETIDINE DERIVATIVES
摘要 Compounds of formula (I) are inhibitors of fatty acid amide hydrolase, (FAAH), and which are useful in the treatment of diseases or medical conditions which benefit from inhibition of FAAH activity, such as anxiety, depression pain, inflammation, and eating, sleep, neurodegenerative and movement disorders: Formula (I) Wherein Ar1 is optionally substituted phenyl or optionally substituted monocyclic heteroaryl having 5 or 6 ring atoms; Ar2 is optionally substituted phenyl, optionally substituted monocyclic heteroaryl having 5 or 6 ring atoms or optionally substituted fused bicyclic heteroaryl having 5 or 6 ring atoms in each fused ring; and Ar3 is a divalent radical selected from the group consisting of optionally substituted phenylene and optionally substituted monocyclic heteroarylene radicals having 5 or 6 ring atoms.
申请公布号 WO2009109743(A1) 申请公布日期 2009.09.11
申请号 WO2009GB00568 申请日期 2009.02.27
申请人 VERNALIS (R&D) LTD.;ROUGHLEY, STEPHEN;WALLS, STEVEN;HART, TERRENCE;PARSONS, RACHEL;BROUGH, PAUL;GRAHAM, CHRISTOPHER;MACIAS, ALBA 发明人 ROUGHLEY, STEPHEN;WALLS, STEVEN;HART, TERRENCE;PARSONS, RACHEL;BROUGH, PAUL;GRAHAM, CHRISTOPHER;MACIAS, ALBA
分类号 C07D205/04;C07D401/12;C07D401/14;C07D413/14 主分类号 C07D205/04
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