发明名称 |
VITAMIN D RECEPTOR MODULATORS |
摘要 |
The present invention relates to novel, non-secosteroidal, diaryl compounds with vitamin D receptor (VDR) modulating activity that are less hypercalcemic than 1a,25 dihydroxy vitamin D3. These compounds are useful for treating bone disease and psoriasis.
|
申请公布号 |
US2009227604(A1) |
申请公布日期 |
2009.09.10 |
申请号 |
US20090470677 |
申请日期 |
2009.05.22 |
申请人 |
BUNEL EMILIO ENRIQUE;GAJEWSKI ROBERT PETER;JONES CHARLES DAVID;LU JIANLIANG;MA TIANWEI;NAGPAL SUNIL;YEE YING KWONG |
发明人 |
BUNEL EMILIO ENRIQUE;GAJEWSKI ROBERT PETER;JONES CHARLES DAVID;LU JIANLIANG;MA TIANWEI;NAGPAL SUNIL;YEE YING KWONG |
分类号 |
A61K31/515;A61P19/10;C07C59/48;C07C59/64;C07C59/66;C07C59/90;C07C65/24;C07C65/34;C07C65/40;C07C69/732;C07C69/734;C07C69/738;C07C69/76;C07C69/94;C07C235/34;C07C235/42;C07C311/51;C07C317/28;C07D207/26;C07D207/27;C07D233/78;C07D239/02;C07D257/04;C07D257/06;C07D261/12;C07D271/10;C07D271/113;C07D277/34;C07D295/185 |
主分类号 |
A61K31/515 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|