发明名称 PIPERAZINE COMPOUNDS, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
摘要 COMPOUND OF FORMULA (1): Y N R2 O-AK-AR R3 X R4 WHEREIN: - RI, R2, R3 AND R4, WHICH MAY BE THE SAME OR DIFFERENT, EACH REPRESENT AN ATOM OR GROUP SELECTED FROM H, HALOGEN, ALKYL, ALKOXY, PHENYL AND CYANO, - X REPRESENTS A BOND, AN OXYGEN ATOM OR A GROUP SELECTED FROM -(CH2)M-, -OCH,- AND -N-R5-, WHEREIN M REPRESENTS 1 OR 2, AND R5 IS AS DEFINED IN THE DESCRIPTION, - Y REPRESENTS AN OXYGEN ATOM OR A GROUP SELECTED FROM NR7 AND CHR8, WHEREIN R7 AND R8 ARE AS DEFINED IN THE DESCRIPTION, - Z REPRESENTS A NITROGEN ATOM OR A CH GROUP, - N REPRESENTS 1 OR 2, - AK REPRESENTS AN ALKYLENE CHAIN,-AR REPRESENTS AN ARYL OR HELEROARYL GROUP, ITS OPTICAL ISOMERS, AND ALSO ADDITION SALTS THEREOF WITH A PHARMACEULICALLY ACCEPTABLE ACID.MEDICAMENTS.
申请公布号 MY139011(A) 申请公布日期 2009.08.28
申请号 MYPI20061556 申请日期 2006.04.06
申请人 LES LABORATOIRES SERVIER 发明人 JEAN-LOUIS PEGLION;AIMEE DESSINGES;BERTRAND GOUMENT;MARK MILLAN;CLOTILDE MANNOURY LA COUR
分类号 C07D313/08;A61P25/00;C07D239/02 主分类号 C07D313/08
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