| 摘要 |
<p>The invention relates to a process for the preparation of anagrelide, and for the preparation of intermediates for use in preparing anagrelide. The invention also relates to the intermediates per se, in particular compounds of Formula (V): where R constitutes a suitable leaving group, which may not be hydrogen. The R group may be selected from: (i)—SiR13, (ii)—CH2Ar, (iii)—COOR2, and (iv) sulfonates such as—SO2R3.</p> |
