| 发明名称 |
PROCESS FOR THE PREPARATION OF 2,3,4,9-TETRAHYDRO-1H-BETA-CARBOLIN-3-CARBOXYLIC ACID ESTERS |
| 摘要 |
<p>The present invention relates to the process of preparation of 2,3,4,9-tetrahydro- 1 /-/-ß-carbolin-3-carboxylic acid esters substituted in position 1 of the general formula (I). in the preferred diastereoisomeric form through a single step starting from tryptophan in racemic form and/or its enantiomers and from 3,4-(methylenedioxy)benzaldehyde.</p> |
| 申请公布号 |
WO2009103787(A1) |
申请公布日期 |
2009.08.27 |
| 申请号 |
WO2009EP52037 |
申请日期 |
2009.02.20 |
| 申请人 |
ENDURA S.P.A.;UNIVERSITA DEGLI STUDI DI FIRENZE;BORZATTA, VALERIO;SCARPI, DINA;GUARNA, ANTONIO;OCCHIATO, ERNESTO |
发明人 |
BORZATTA, VALERIO;SCARPI, DINA;GUARNA, ANTONIO;OCCHIATO, ERNESTO |
| 分类号 |
C07D471/04 |
主分类号 |
C07D471/04 |
| 代理机构 |
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