发明名称 4, 5-DIHYDRO-OXAZOL-2-YL AMINE DERIVATIVES
摘要 The present invention relates to a compounds of formula I or a pharmaceutically active acid addition salts thereof. It has been found that the present compounds have Asp2 (ß-sccretasc, BACE 1 or Mcmapsin-2) inhibitory activity and that the compounds may therefore be used in the treatment of diseases characterised by elevated ß-amyloid levels or ß-amyloid deposits, particularly Alzheimer's disease.
申请公布号 WO2009103626(A1) 申请公布日期 2009.08.27
申请号 WO2009EP51452 申请日期 2009.02.09
申请人 F. HOFFMANN-LA ROCHE AG;SIENA BIOTECH S.P.A;ANDREINI, MATTEO;GABELLIERI, EMANUELE;GUBA, WOLFGANG;MARCONI, GUIDO;NARQUIZIAN, ROBERT;POWER, EOIN;TRAVAGLI, MASSIMILIANO;WOLTERING, THOMAS;WOSTL, WOLFGANG 发明人 ANDREINI, MATTEO;GABELLIERI, EMANUELE;GUBA, WOLFGANG;MARCONI, GUIDO;NARQUIZIAN, ROBERT;POWER, EOIN;TRAVAGLI, MASSIMILIANO;WOLTERING, THOMAS;WOSTL, WOLFGANG
分类号 C07D263/28;A61K31/422;A61P25/28;C07D413/10 主分类号 C07D263/28
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