发明名称 BICYCLOAMINE DERIVATIVE
摘要 <p>Disclosed is a compound represented by Formula (I) or a pharmaceutically acceptable salt thereof, which has an excellent inhibitory activity on a sodium channel and is therefore useful as a therapeutic agent for various types of neuralgia, nervous disorders, epilepsy, insomnia, premature ejaculation and others or as an analgesic agent. (I) wherein Q represents an ethylene or the like; R1, R2 and R3 independently represent a hydrogen or the like; X1 represents a C1-6 alkylene or the like; X2 represents a C1-6 alkylene or the like; A1 represent a 5- to 6-membered heterocyclic group or the like; and A2 represents a C6-14 aryl or the like.</p>
申请公布号 WO2009101917(A1) 申请公布日期 2009.08.20
申请号 WO2009JP52164 申请日期 2009.02.09
申请人 EISAI R & D MANAGEMENT CO., LTD.;OZAKI, FUMIHIRO;SOEJIMA, MOTOHIRO;ISHIDA, TASUKU;NORIMINE, YOSHIHIKO;KURUSU, NOBUYUKI;DOI, ERIKO;KANEKO, TOSHIHIKO;HASEGAWA, DAIJU;KOBAYASHI, KIYOAKI;YAMAMOTO, NOBORU 发明人 OZAKI, FUMIHIRO;SOEJIMA, MOTOHIRO;ISHIDA, TASUKU;NORIMINE, YOSHIHIKO;KURUSU, NOBUYUKI;DOI, ERIKO;KANEKO, TOSHIHIKO;HASEGAWA, DAIJU;KOBAYASHI, KIYOAKI;YAMAMOTO, NOBORU
分类号 C07D451/06;A61K31/439;A61K31/46;A61K31/4985;A61K31/53;A61K31/5377;A61K31/5383;A61K31/55;A61P3/12;A61P15/00;A61P25/00;A61P25/04;A61P25/08;A61P25/20;A61P29/02;A61P43/00;C07D451/14;C07D519/00 主分类号 C07D451/06
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