发明名称 THE HEMI-FUMARATE SALT OF A 1,3,4-THIADIAZOLYL DERIVATIVE AS MODULATOR OF THE SPHINGOSINE 1-PHOSPHATE RECEPTOR
摘要 <p>The invention relates to the compound (2S)-2-amino-2-{5-[4-(octyloxy)-3- (trifluoromethyl)phenyl]-1,3,4-thiadiazol-2-yl}-1-propanol hemi-fumarate, processes for its preparation, pharmaceutical compositions containing them and its use in the treatment of conditions or disorders which are mediated via the S1 P1 receptor.</p>
申请公布号 WO2009098193(A1) 申请公布日期 2009.08.13
申请号 WO2009EP51175 申请日期 2009.02.03
申请人 GLAXO GROUP LIMITED;ANSON, MICHAEL, SIMON;DAY, CAROLINE, JANE;GRAHAM, JONATHAN, PAUL;KINDON, LEANDA, JANE;WOOLLAM, GRAHAME, ROBERT 发明人 ANSON, MICHAEL, SIMON;DAY, CAROLINE, JANE;GRAHAM, JONATHAN, PAUL;KINDON, LEANDA, JANE;WOOLLAM, GRAHAME, ROBERT
分类号 C07D277/28;A61K31/433;A61P25/00 主分类号 C07D277/28
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