发明名称 |
TRICYCLIC COMPOUNDS HAVING CORTICOTROPIN-RELEASING FACTOR ANTAGONISTIC ACTIVITY AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
摘要 |
<p>There is provided a compound of the formula (I') : wherein X is a nitrogen or CRx, Rx is a hydrogen, etc., R1 is an optionally substituted hydrocarbon group, etc., R2 is an optionally substituted hydrocarbon group, etc., ring A is 5- to -8-membered heterocyclic ring, etc., and each of Y1,. Y2 and Y3 is an optionally substituted carbon or a nitrogen, etc.; or 'a salt thereof or a prodrug thereof., which have CRF receptor antagonistic activity and use thereof.</p> |
申请公布号 |
WO2009093747(A1) |
申请公布日期 |
2009.07.30 |
申请号 |
WO2009JP51299 |
申请日期 |
2009.01.21 |
申请人 |
TAKEDA PHARMACEUTICAL COMPANY LIMITED;ASO, KAZUYOSHI;KOBAYASHI, KATSUMI;TAKAI, TAKAFUMI;KOJIMA, TAKUTO;TOKUMARU, KAZUYUKI;MOCHIZUKI, MICHIYO;HOASHI, YASUTAKA |
发明人 |
ASO, KAZUYOSHI;KOBAYASHI, KATSUMI;TAKAI, TAKAFUMI;KOJIMA, TAKUTO;TOKUMARU, KAZUYUKI;MOCHIZUKI, MICHIYO;HOASHI, YASUTAKA |
分类号 |
C07D487/04;A61K31/4188;A61P25/22;A61P25/24;C07D498/04 |
主分类号 |
C07D487/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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