发明名称 TRICYCLIC COMPOUNDS HAVING CORTICOTROPIN-RELEASING FACTOR ANTAGONISTIC ACTIVITY AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
摘要 <p>There is provided a compound of the formula (I') : wherein X is a nitrogen or CRx, Rx is a hydrogen, etc., R1 is an optionally substituted hydrocarbon group, etc., R2 is an optionally substituted hydrocarbon group, etc., ring A is 5- to -8-membered heterocyclic ring, etc., and each of Y1,. Y2 and Y3 is an optionally substituted carbon or a nitrogen, etc.; or 'a salt thereof or a prodrug thereof., which have CRF receptor antagonistic activity and use thereof.</p>
申请公布号 WO2009093747(A1) 申请公布日期 2009.07.30
申请号 WO2009JP51299 申请日期 2009.01.21
申请人 TAKEDA PHARMACEUTICAL COMPANY LIMITED;ASO, KAZUYOSHI;KOBAYASHI, KATSUMI;TAKAI, TAKAFUMI;KOJIMA, TAKUTO;TOKUMARU, KAZUYUKI;MOCHIZUKI, MICHIYO;HOASHI, YASUTAKA 发明人 ASO, KAZUYOSHI;KOBAYASHI, KATSUMI;TAKAI, TAKAFUMI;KOJIMA, TAKUTO;TOKUMARU, KAZUYUKI;MOCHIZUKI, MICHIYO;HOASHI, YASUTAKA
分类号 C07D487/04;A61K31/4188;A61P25/22;A61P25/24;C07D498/04 主分类号 C07D487/04
代理机构 代理人
主权项
地址