发明名称 ALDH-2 INHIBITORS IN THE TREATMENT OF ADDICTION
摘要 Disclosed are novel isoflavone derivatives having the structure of Formula I which are useful as ALDH-2 inhibitors for treating mammals for dependence upon drugs of addiction, for example addiction to dopamine-producing agent such as cocaine, morphine, amphetamines, nicotine, and alcohol.
申请公布号 CA2712750(A1) 申请公布日期 2009.07.30
申请号 CA20082712750 申请日期 2008.01.24
申请人 GILEAD PALO ALTO, INC.;THE ENDOWMENT FOR RESEARCH IN HUMAN BIOLOGY, INC. 发明人 BILOKIN, YAROSLAV;ELZEIN, ELFATIH;ZABLOCKI, JEFF;ORGAN, MICHAEL;PERRY, THAO;KOBAYASHI, TETSUYA;ABELMAN, MATTHEW;KALLA, RAO;FAN, PEIDONG;DIAMOND, IVAN;JIANG, ROBERT;AROLFO, MARIA PIA;LI, XIAOFEN;YAO, LINA;JIANG, ZHAN;KEUNG, WING MING;TAO, GUOXIN
分类号 C07D311/36;A61K31/353;A61P25/32;C07D405/04;C07D405/14;C07D413/12;C07D413/14;C07D417/12 主分类号 C07D311/36
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