发明名称 IMPROVED PROCESS FOR THE PREPARATION OF (S)-PREGABALIN
摘要 The present invention provides a process for resolving racemic pregabalin to S-pregabalin by using a chiral acid to form a pregabalin salt, purifying the salt to obtain a purified S-pregabalin salt then neutralizing the salt to obtain S-pregabalin having good chiral purity.
申请公布号 WO2009087674(A2) 申请公布日期 2009.07.16
申请号 WO2008IN00845 申请日期 2008.12.18
申请人 WATSON PHARMA PRIVATE LIMITED;CHAVAN, AMIT, ANANT;PADWAL, SHASHIKANT, BALASAHEB;JOSHI, ASHUTOSH, VIJAY;BHANU, MANJUNATH, NARAYAN 发明人 CHAVAN, AMIT, ANANT;PADWAL, SHASHIKANT, BALASAHEB;JOSHI, ASHUTOSH, VIJAY;BHANU, MANJUNATH, NARAYAN
分类号 C07C227/34;C07C227/40 主分类号 C07C227/34
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