发明名称 |
STREPTOGRAMIN DERIVATIVE, PREPARATION THEREOF AND COMPOSITION CONTAINING THE SAME |
摘要 |
PROBLEM TO BE SOLVED: To provide a novel antibacterial agent with advantageous antibacterial activity. SOLUTION: Group A streptogramin derivatives is expressed by general formula (I), wherein: R<SB>1</SB>represents cyano or ethynyl radicals; R<SB>2</SB>represents a hydrogen atom or a methyl or ethyl radical; and a bond of formula (α) represents a single bond (stereochemistry 27R) or a double bond. COPYRIGHT: (C)2009,JPO&INPIT
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申请公布号 |
JP2009149627(A) |
申请公布日期 |
2009.07.09 |
申请号 |
JP20080302750 |
申请日期 |
2008.11.27 |
申请人 |
NOVEXEL |
发明人 |
DESMAZEAU PASCAL;RONAN BAPTISTE;BACQUE ERIC;BARRIERE JEAN-CLAUDE |
分类号 |
A61K31/424;C07D498/14;A61K31/42;A61K31/444;A61K38/00;A61P31/04;A61P43/00;C07D498/16;C07D498/18;C07D498/22;C07K5/06;C07K5/078 |
主分类号 |
A61K31/424 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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