发明名称 NOVEL PROCESS FOR SYNTHESIS OF ITOPRIDE AND ITS NOVEL INTERMEDIATE N-(4-HYDROXYBENZYL)- 3,4-DIMETHOXYBENZAMIDE
摘要 The present invention relates to a novel and improved process for the preparation of N-[4-[2-(dimethylamino)ethoxy]benzyl]-3,4-dimethoxybenzamide-known as Itopride, via a novel intermediate N-(4~hydroxybenzyl)-3,4-dimethoxybenzamide.
申请公布号 US2009177008(A1) 申请公布日期 2009.07.09
申请号 US20060159291 申请日期 2006.12.28
申请人 CADILA PHARMACEUTICALS LTD. 发明人 KHAMAR BAKULESH MAFATLAL;MODI INDRAVADAN AMBALAL;VENKATRAMAN JAYARAMAN;RAVI PONNAIAH;NORI DIVAKARA SOMAYAJULU;GAJULA MADHUSUDANA RAO;RENUGADEVI GURUSAMY;SHASHIKALA KUNJARU N.;RUDRAMUNI SANTOSH M.
分类号 C07C231/10;C07C233/60 主分类号 C07C231/10
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