IMPROVED PROCESS FOR THE PREPARATION OF (1-BENZYL-4-(5,6,- DIMETHOXYIND ANONE-2-YL)METHYLPIPERIDINE) HYDROCHLORIDE-FORM III
摘要
The present invention is directed to an improved industrially viable, cost effective process for manufacturing pure racemic crystalline anhydrous form of (1-benzyl-4-(5,6,- dimethoxyindanone-2yl)methylpiperidine) hydrochloride Form III commonly known as Donepezil hydrochloride with a purity level of greater than 99.9%.
申请公布号
WO2009084030(A2)
申请公布日期
2009.07.09
申请号
WO2008IN00805
申请日期
2008.12.02
申请人
NEULAND LABORATORIES LTD.;RAMAKRISHNAN, ARUL;BATHANI, GURUSWAMY;BANDARI, HARIBABU;GOPU, RAVI SHANKAR
发明人
RAMAKRISHNAN, ARUL;BATHANI, GURUSWAMY;BANDARI, HARIBABU;GOPU, RAVI SHANKAR