发明名称 IMPROVED PROCESS FOR THE PREPARATION OF (1-BENZYL-4-(5,6,- DIMETHOXYIND ANONE-2-YL)METHYLPIPERIDINE) HYDROCHLORIDE-FORM III
摘要 The present invention is directed to an improved industrially viable, cost effective process for manufacturing pure racemic crystalline anhydrous form of (1-benzyl-4-(5,6,- dimethoxyindanone-2yl)methylpiperidine) hydrochloride Form III commonly known as Donepezil hydrochloride with a purity level of greater than 99.9%.
申请公布号 WO2009084030(A2) 申请公布日期 2009.07.09
申请号 WO2008IN00805 申请日期 2008.12.02
申请人 NEULAND LABORATORIES LTD.;RAMAKRISHNAN, ARUL;BATHANI, GURUSWAMY;BANDARI, HARIBABU;GOPU, RAVI SHANKAR 发明人 RAMAKRISHNAN, ARUL;BATHANI, GURUSWAMY;BANDARI, HARIBABU;GOPU, RAVI SHANKAR
分类号 C07D211/32;C07C49/633 主分类号 C07D211/32
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