发明名称 PROCESS FOR PRODUCTION OF 4-(SUBSTITUTED PHENYL)HEXAHYDROPYRIDO[2,1-C][1,4]OXAZIN-6-ONE
摘要 <p>4-(Substituted phenyl)hexahydropyrido[2,1-c][1,4]oxazin- 6-one represented by formula (I) or a salt thereof is useful as an intermediate for the production of a bicyclic cinnamide compound which is an Aß production inhibitor. 4-(Substituted phenyl)hexahydropyrido[2,1-c][1,4]oxazin-6-one or the salt thereof can be produced in an industrially advantageous manner by subjecting a compound represented by formula (II) or a salt thereof to an intramolecular condensation reaction.</p>
申请公布号 WO2009081959(A1) 申请公布日期 2009.07.02
申请号 WO2008JP73513 申请日期 2008.12.25
申请人 EISAI R & D MANAGEMENT CO., LTD.;KAYANO, AKIO;NAGAI, MITSUO;HOSHINO, YORIHISA;WAKASUGI, KAZUNORI;MATSUDA, MASAAKI;KAMADA, ATSUSHI;ISOMURA, MINETAKA;NISHIKAWA, YOSHIHIRO;YOSHIKAWA, SEIJI;SHIMMYO, DAISUKE;DOI, ERIKO;KANEKO, TOSHIHIKO 发明人 KAYANO, AKIO;NAGAI, MITSUO;HOSHINO, YORIHISA;WAKASUGI, KAZUNORI;MATSUDA, MASAAKI;KAMADA, ATSUSHI;ISOMURA, MINETAKA;NISHIKAWA, YOSHIHIRO;YOSHIKAWA, SEIJI;SHIMMYO, DAISUKE;DOI, ERIKO;KANEKO, TOSHIHIKO
分类号 C07D498/04;C07D265/30 主分类号 C07D498/04
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